Flupirtine

3 Topics Found

FLUDOL (Flupirtine) is a centrally acting, non-opioid analgesic that is available in a number of European countries for the treatment of a variety of pain states. The therapeutic benefits seen with flupirtine relate to its unique pharmacological properties. FLUDOL (Flupirtine) displays indirect NDMA receptor antagonism via activation of potassium channels and is the first representative of a pharmacological class denoted the ‘selective neuronal potassium channel openers’. The generation of the M-current is facilitated by flupirtine via the opening of neuronal Kv7 potassium channels. The opening of these channels inhibits exaggerated neuronal action potential generation and controls neuronal excitability. Neuronal hyperexcitability is a physiological ...

Filed under Tramadol

Flupirtine is a centrally acting, non-opioid analgesic that is available in a number of European countries for the treatment of a variety of pain states. The therapeutic benefits seen with flupirtine relate to its unique pharmacological properties. Flupirtine displays indirect NDMA receptor antagonism via activation of potassium channels and is the first representative of a pharmacological class denoted the ‘selective neuronal potassium channel openers’. The generation of the M-current is facilitated by flupirtine via the opening of neuronal Kv7 potassium channels. The opening of these channels inhibits exaggerated neuronal action potential generation and controls neuronal excitability. Neuronal hyperexcitability is a physiological component of many ...

1 REPLY Filed under Tramadol

is lupins katadol caps harmless in case of kideny stones ? ## I have a problem of heart pain went to doc they pescrib me these tablets but after sm time it unable to relif me from my pain. What should I do the pain is giving me hell of a pain. ## Please reffer me some medicens name which can reliff me from heart pain its not heart attack. Im using Lupkin's Katadol Caps 3.5gm. ## @neelam, Based on my research there are no interactions or contraindications listed between Lupin Katadol (Flupirtine maleate) and those with kidney stones. I can't say whether or not it's harmless, as every individual may react differently. But from what I've read, it's not likely that you'd experience any problems on that end. @Nisha, If the medication you're using isn't working...

4 REPLIES Filed under Codeine

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