Antagon

Ganirelix

Ganirelix acetate (or diacetate), sold under the brand names Orgalutran and Antagon among others, is an injectable competitive gonadotropin-releasing hormone antagonist (GnRH antagonist). It is primarily used in assisted reproduction to control ovulation. The drug works by blocking the action of GnRH upon the pituitary, thus rapidly suppressing the production and action of LH and FSH. Ganirelix is used in fertility treatment to prevent premature ovulation that could result in the harvesting ...

do you know which would be the safest selective 5ht2b antagonist there is to prevent cardiac fibrosis in terms of physical damage. i am looking for one to take with certain anti depressants that are 5ht2b agonists and have been shown to cause valvular fibrosis. i am looking for one selective to 5ht2b.

I have been taking inj.Tramadol 800 mg as two decided injections.Thogh the buzz associated with this is absent for quite some time any small irritation make me go for Tramadol. I am in a job I detested and still I am in the same job I hate. Plenty of opportunity to go back to Tramadol . Someone recently said I could take Nexito that would stop the craving .

Prescription of zandip 20 mg , physiotens 0.4mg, karvezide 300 mg for high b.p ( 180/80). Recently added verpamil hydrochloride SR 240 mg trial with 0.4 mg physiotens, karvezide and Zanadip 10 mg. is this combo compatible? There is not much improvement. ## Are you also watching your diet? If you're sodium sensitive, then that could cause blood pressure elevation. Do you also get lots of proper exercise? That is also vital to blood pressure control. You really can't just take medications and expect them to do all of the work. What types of foods do you normally eat? Do you have any other medical conditions?

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Tecastemizole

H1 antagonists, also called H1 blockers, are a class of medications that block the action of histamine at the H1 receptor, helping to relieve allergic reactions. Agents where the main therapeutic effect is mediated by negative modulation of histamine receptors are termed antihistamines; other agents may have antihistaminergic action but are not true antihistamines.[citation needed] In common use, the term "antihistamine" refers only to H1-antihistamines. Virtually all H1-anti...

Drug Index

H1 antagonists, also called H1 blockers, are a class of medications that block the action of histamine at the H1 receptor, helping to relieve allergic reactions. Agents where the main therapeutic effect is mediated by negative modulation of histamine receptors are termed antihistamines; other agents may have antihistaminergic action but are not true antihistamines.[citation needed] In common use, the term "antihistamine" refers only to H1-antihistamines. Virtually all H1-anti...

Cyclopentolate

Cyclopentolate is a muscarinic antagonist.[1] It is commonly used as an eye drop during pediatric eye examinations to dilate the eye (mydriatic) and prevent the eye from focusing/accommodating (cycloplegic). Cyclopentolate or atropine can also be administered to reverse muscarinic and central nervous system effects of indirect cholinomimetic (anti-AChase) administration. It is on the World Health Organization's List of Essential Medicines.[2] After instillatio...

Cyclopentolate

Cyclopentolate is a muscarinic antagonist.[1] It is commonly used as an eye drop during pediatric eye examinations to dilate the eye (mydriatic) and prevent the eye from focusing/accommodating (cycloplegic). Cyclopentolate or atropine can also be administered to reverse muscarinic and central nervous system effects of indirect cholinomimetic (anti-AChase) administration. It is on the World Health Organization's List of Essential Medicines.[2] After instillatio...

Nizatidine

Nizatidine is a histamine H2 receptor antagonist that inhibits stomach acid production, and is commonly used in the treatment of peptic ulcer disease and gastroesophageal reflux disease.[1] It was patented in 1980 and approved for medical use in 1988.[2][3] It was developed by Eli Lilly. Brand names include Tazac and Axid. Contents 1 Medical use 2 Adverse effects 3 History and development 4 See also 5 References 6 External links Medical u...

Cyclopentolate + Phenylephrine

Cyclopentolate is a muscarinic antagonist.[1] It is commonly used as an eye drop during pediatric eye examinations to dilate the eye (mydriatic) and prevent the eye from focusing/accommodating (cycloplegic). Cyclopentolate or atropine can also be administered to reverse muscarinic and central nervous system effects of indirect cholinomimetic (anti-AChase) administration. It is on the World Health Organization's List of Essential Medicines.[2] After instillatio...

Cyclopentolate

Cyclopentolate is a muscarinic antagonist.[1] It is commonly used as an eye drop during pediatric eye examinations to dilate the eye (mydriatic) and prevent the eye from focusing/accommodating (cycloplegic). Cyclopentolate or atropine can also be administered to reverse muscarinic and central nervous system effects of indirect cholinomimetic (anti-AChase) administration. It is on the World Health Organization's List of Essential Medicines.[2] After instillatio...

Drug Index

Cyclopentolate is a muscarinic antagonist.[1] It is commonly used as an eye drop during pediatric eye examinations to dilate the eye (mydriatic) and prevent the eye from focusing/accommodating (cycloplegic). Cyclopentolate or atropine can also be administered to reverse muscarinic and central nervous system effects of indirect cholinomimetic (anti-AChase) administration. It is on the World Health Organization's List of Essential Medicines.[2] After instillatio...

Azilsartan Medoxomil

Azilsartan is an angiotensin II receptor antagonist used in the treatment of hypertension,[1][2][3] developed by Takeda. It is marketed in tablet form under the brand name Edarbi as the prodrug azilsartan medoxomil.[4] The most common adverse reaction in adults is diarrhea.[1] It is also sold as a combination drug with chlortalidone under the brand name Edarbyclor.[5] Contents 1 Structure activit...

Granisetron

Granisetron is a serotonin 5-HT3 receptor antagonist used as an antiemetic to treat nausea and vomiting following chemotherapy and radiotherapy. Its main effect is to reduce the activity of the vagus nerve, which is a nerve that activates the vomiting center in the medulla oblongata. It does not have much effect on vomiting due to motion sickness. This drug does not have any effect on dopamine receptors or muscarinic receptors. Granisetron was developed by chemists working at the British dr...

Drug Index

Nizatidine is a histamine H2 receptor antagonist that inhibits stomach acid production, and is commonly used in the treatment of peptic ulcer disease and gastroesophageal reflux disease.[1] It was patented in 1980 and approved for medical use in 1988.[2][3] It was developed by Eli Lilly. Brand names include Tazac and Axid. Contents 1 Medical use 2 Adverse effects 3 History and development 4 See also 5 References 6 External links Medical u...

Granisetron

Granisetron is a serotonin 5-HT3 receptor antagonist used as an antiemetic to treat nausea and vomiting following chemotherapy and radiotherapy. Its main effect is to reduce the activity of the vagus nerve, which is a nerve that activates the vomiting center in the medulla oblongata. It does not have much effect on vomiting due to motion sickness. This drug does not have any effect on dopamine receptors or muscarinic receptors. Granisetron was developed by chemists working at the British dr...

Eprosartan

Eprosartan is an angiotensin II receptor antagonist used for the treatment of high blood pressure. It is marketed in the United States as Teveten by Abbvie, the spin-off of the pharmaceutical discovery division of Abbott Laboratories; it is marketed as Eprozar by Intas Pharmaceuticals in India, and by Abbott Laboratories elsewhere. The compound came into the Abbott Laboratories cardiovascular pipeline with its acquisition of Kos Pharmaceuticals in 2006, which had licensed it, along with "a ra...

Granisetron

Granisetron is a serotonin 5-HT3 receptor antagonist used as an antiemetic to treat nausea and vomiting following chemotherapy and radiotherapy. Its main effect is to reduce the activity of the vagus nerve, which is a nerve that activates the vomiting center in the medulla oblongata. It does not have much effect on vomiting due to motion sickness. This drug does not have any effect on dopamine receptors or muscarinic receptors. Granisetron was developed by chemists working at the British dr...

Abciximab

Abciximab, a glycoprotein IIb/IIIa receptor antagonist manufactured by Janssen Biologics BV and distributed by Eli Lilly under the trade name ReoPro, is a platelet aggregation inhibitor mainly used during and after coronary artery procedures like angioplasty to prevent platelets from sticking together and causing thrombus (blood clot) formation within the coronary artery. It is a glycoprotein IIb/IIIa inhibitor.[3] While abciximab has a short plasma half-life, due to its stron...

Azilsartan Medoxomil + Chlorthalidone

Azilsartan is an angiotensin II receptor antagonist used in the treatment of hypertension,[1][2][3] developed by Takeda. It is marketed in tablet form under the brand name Edarbi as the prodrug azilsartan medoxomil.[4] The most common adverse reaction in adults is diarrhea.[1] It is also sold as a combination drug with chlortalidone under the brand name Edarbyclor.[5] Contents 1 Structure activit...