Macitentan

Category: Blood Pressure

Macitentan Overview

Macitentan, sold under the brand name Opsumit, is an endothelin receptor antagonist (ERA) approved for the treatment of pulmonary arterial hypertension (PAH).[2] The other two ERAs marketed as of 2014 are bosentan and ambrisentan.[2] Macitentan is a dual ERA, meaning that it acts as an antagonist of two endothelin (ET) receptor subtypes, ETA and ETB.[2] However, macitentan has a 50-fold increased selectivity for the ETA subtype compared to the E...

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Details May Include Instructions, Side Effects, Interactions, Etc. Drug monograph is from Wikipedia. All text is available under the terms of the GFDL (GNU Free Documentation License). Source: en.wikipedia.org/wiki/Macitentan

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Other drugs which contain Macitentan or a similar ingredient: (1 result)

• OPSUMIT Macitentan